F. DA SETTIMO: search on Z-Library

The world's largest scientific articles store. 70,000,000+ articles for free.

Don't use scam websites

1

Geometrically Constrained Derivatives of Indolylglyoxylamides as Ligands Binding the GABAA/BzR Complex

Sartini, S., Morelli, M., Simorini, F., Taliani, S., Salerno, S., M. Marini, A., Da Settimo, F., La Motta, C.

Journal:

Current Topics in Medicinal Chemistry

Year:

2012

Language:

english

File:

PDF, 494 KB

english, 2012

2

Structural Requirements to Obtain Highly Potent and Selective 18 kDa Translocator Protein (TSPO) Ligands

Taliani, Sabrina, Pugliesi, Isabella, Da Settimo, Federico

Journal:

Current Topics in Medicinal Chemistry

Year:

2011

Language:

english

File:

PDF, 492 KB

english, 2011

3

Targeting the 18-kDa translocator protein: recent perspectives for neuroprotection

Da Pozzo, Eleonora, Giacomelli, Chiara, Barresi, Elisabetta, Costa, Barbara, Taliani, Sabrina, Passetti, Federico Da Settimo, Martini, Claudia

Journal:

Biochemical Society Transactions

Year:

2015

Language:

english

File:

PDF, 246 KB

english, 2015

4

Unbinding of Translocator Protein 18 kDa (TSPO) ligands: from in vitro residence time to in vivo efficacy via in silico simulations

Bruno, Agostino, Barresi, Elisabetta, Simola, Nicola, Da Pozzo, Eleonora, Costa, Barbara, Novellino, Ettore, Da Settimo, Federico, Martini, Claudia, Taliani, Sabrina, Cosconati, Sandro

Journal:

ACS Chemical Neuroscience

Year:

2019

Language:

english

File:

PDF, 942 KB

english, 2019

5

Novel positive allosteric modulators of A 2B adenosine receptor acting as bone mineralisation promoters

Barresi, Elisabetta, Giacomelli, Chiara, Marchetti, Laura, Baglini, Emma, Salerno, Silvia, Greco, Giovanni, Da Settimo, Federico, Martini, Claudia, Trincavelli, Maria Letizia, Taliani, Sabrina

Journal:

Journal of Enzyme Inhibition and Medicinal Chemistry

Year:

2021

File:

PDF, 2.41 MB

2021

6

Geometrically Constrained Analogues of N-Benzylindolylglyoxylylamides: [1, 2, 4]Triazino[4, 3-a]benzimidazol-4(10H)-one Derivatives as Potential New Ligands at the Benzodiazepine Receptor

Giampaolo Primofiore, Federico Da Settimo, Sabrina Taliani, Anna Maria Marini, Francesca Simorini, Ettore Novellino, Giovanni Greco, Letizia Trincavelli, Claudia Martini

Journal:

Archiv der Pharmazie

Year:

2003

Language:

english

File:

PDF, 126 KB

english, 2003

7

Synthesis and Benzodiazepine Receptor Affinity of Derivatives of the New Tricyclic Heteroaromatic System Pyrido[3′,2′:5,6]thiopyrano[4,3-c]pyridazin-3(2H,5H)-one

Giampaolo Primofiore, Federico Da Settimo, Anna Maria Marini, Francesca Simorini, Concettina La Motta, Sabrina Taliani, Sonia Laneri, Letizia Trincavelli, Claudia Martini

Journal:

Archiv der Pharmazie

Year:

2005

Language:

english

File:

PDF, 125 KB

english, 2005

8

Synthesis and Biological Evaluation of 2′-Oxo-2,3-dihydro-3′H- spiro[chromene-4,5′-[1,3]oxazolidin]-3′yl]acetic Acid Derivatives as Aldose Reductase Inhibitors

Simona Rapposelli, Federico Da Settimo, Maria Digiacomo, Concettina La Motta, Annalina Lapucci, Stefania Sartini, Michael Vanni

Journal:

Archiv der Pharmazie

Year:

2011

Language:

english

File:

PDF, 254 KB

english, 2011

9

ChemInform Abstract: Synthesis, Structure-Activity Relationships, and Molecular Modeling Studies of N-(Indol-3-ylglyoxylyl)benzylamine Derivatives Acting at the Benzodiazepine Receptor.

A. DA SETTIMO, G. PRIMOFIORE, F. DA SETTIMO, A. M. MARINI, E. NOVELLINO, G. GRECO, C. MARTINI, G. GIANNACCINI, A. LUCACCHINI

Journal:

Year:

1997

File:

PDF, 30 KB

1997

10

ChemInform Abstract: Benzisothiazole-1,1-dioxide Alkanoic Acid Derivatives as Inhibitors of Rat Lens Aldose Reductase.

G. PRIMOFIORE, F. DA SETTIMO, C. LA MOTTA, F. SIMORINI, A. MINUTOLO

Journal:

Year:

1998

File:

PDF, 26 KB

1998

11

ChemInform Abstract: Synthesis of Purinobenzothiazine and Pyridothiazinopurine Derivatives. Two New Heterocyclic Ring Systems.

A. DA SETTIMO, A. M. MARINI, G. PRIMOFIORE, F. DA SETTIMO, D. BERTINI

Journal:

Year:

1998

File:

PDF, 32 KB

1998

12

ChemInform Abstract: Synthesis, DNA Binding and in vitro Antiproliferative Activity of Purinoquinazoline, Pyridopyrimidopurine and Pyridopyrimidobenzimidazole Derivatives as Potential Antitumor Agents.

A. DA SETTIMO, F. DA SETTIMO, A. M. MARINI, G. PRIMOFIORE, S. SALERNO, G. VIOLA, L. DALLA VIA, S. MARCIANI MAGNO

Journal:

Year:

1999

File:

PDF, 31 KB

1999

13

ChemInform Abstract: Indole Amide Derivatives: Synthesis, Structure—Activity Relationships, and Molecular Modeling Studies of a New Series of Histamine H1-Receptor Antagonists.

Sandra Battaglia, Enrico Boldrini, Federico Da Settimo, Giulio Dondio, Concettina La Motta, Anna Maria Marini, Giampaolo Primofiore

Journal:

Year:

1999

File:

PDF, 31 KB

1999

14

ChemInform Abstract: Synthesis of Purinobenzodiazepine and Purinobenzotriazocine Derivatives, Two New Heterocyclic Ring Systems.

Antonio Da Settimo, Giampaolo Primofiore, Anna Maria Marini, Federico Da Settimo, Concettina La Motta, Silvia Salerno

Journal:

Year:

1999

File:

PDF, 31 KB

1999

15

ChemInform Abstract: 3-Aryl-[1,2,4]triazino[4,3-a]benzimidazol-4(10H)-ones: Tricyclic Heteroaromatic Derivatives as a New Class of Benzodiazepine Receptor Ligands.

Giampaolo Primofiore, Federico Da Settimo, Sabrina Taliani, Anna Maria Marini, Concettina La Motta, Ettore Novellino, Giovanni Greco, Marco Gesi, Letizia Trincavelli, Claudia Martini

Journal:

Year:

2000

Language:

english

File:

PDF, 31 KB

english, 2000

16

ChemInform Abstract: Synthesis of Novel 5H,11H-Pyrido[2′,3′:2,3]thiopyrano[4,3-b]indoles by Fischer-Indole Cyclization.

Antonio Da Settimo, Anna Maria Marini, Giampaolo Primofiore, Federico Da Settimo, Silvia Salerno, Concettina La Motta, Gianluca Pardi, Pier Luigi Ferrarini, Claudio Mori

Journal:

Year:

2000

File:

PDF, 30 KB

2000

17

ChemInform Abstract: Synthesis of a Novel Purine-Containing Heterocyclic Ring System: 8,10-Dimethylindolo[2′,3′:5,6][1,2,4]triazino [4,3-f]purine-9,11(8H,10H,13H)-dione.

Antonio Da Settimo, Giampaolo Primofiore, Federico Da Settimo, Francesca Simorini, Anna Maria Marini, Concettina La Motta, Sabrina Taliani

Journal:

Year:

2000

File:

PDF, 33 KB

2000

18

ChemInform Abstract: 3-Aryl[1,2,4]triazino[4,3-a]benzimidazol-4(10H)-ones: A New Class of Selective A1 Adenosine Receptor Antagonists.

Federico Da Settimo, Giampaolo Primofiore, Sabrina Taliani, Anna Maria Marini, Concettina La Motta, Ettore Novellino, Giovanni Greco, Antonio Lavecchia, Letizia Trincavelli, Claudia Martini

Journal:

Year:

2001

File:

PDF, 33 KB

2001

19

ChemInform Abstract: Synthesis, in vitro Antiproliferative Activity and DNA-Interaction of Benzimidazoquinazoline Derivatives as Potential Antitumor Agents.

Lisa Dalla Via, Ornella Gia, Sebastiano Marciani Magno, Antonio Da Settimo, Anna Maria Marini, Giampaolo Primofiore, Frederico Da Settimo, Silvia Salerno

Journal:

Year:

2001

File:

PDF, 29 KB

2001

20

ChemInform Abstract: Facile Synthesis of 3-Substituted [1,2,4]Triazino[3,4-f]purine-4,6,8-trione Derivatives.

Federico Da Settimo, Anna Maria Marini, Gianluca Pardi, Giampaolo Primofiore, Silvia Salerno, Francesca Simorini

Journal:

Year:

2001

File:

PDF, 30 KB

2001

21

ChemInform Abstract: [1,2,4]Triazino[4,3-a]benzimidazole Acetic Acid Derivatives: A New Class of Selective Aldose Reductase Inhibitors.

Federico Da Settimo, Giampaolo Primofiore, Antonio Da Settimo, Concettina La Motta, Sabrina Taliani, Francesca Simorini, Ettore Novellino, Giovanni Greco, Antonio Lavecchia, Enrico Boldrini

Journal:

Year:

2002

File:

PDF, 31 KB

2002

22

Dialkylaminoalkylindolonaphthyridines as Potential Antitumor Agents: Synthesis, Cytotoxicity and DNA Binding Properties.

Lisa Dalla Via, Ornella Gia, Sebastiano Marciani Magno, Antonio Da Settimo, Giampaolo Primofiore, Federico Da Settimo, Francesca Simorini, Anna Maria Marini

Journal:

Year:

2002

File:

PDF, 32 KB

2002

23

Synthesis of Novel Pyrido[3′,2′:5,6]thiopyrano[3,2-b]indol-5(6H)-ones and 6H-Pyrido[3′,2′:5,6]thiopyrano[4,3-b]quinolines, Two New Heterocyclic Ring Systems.

Antonio Da Settimo, Anna Maria Marini, Giampaolo Primofiore, Federico Da Settimo, Silvia Salerno, Francesca Simorini, Gianluca Pardi, Concettina La Motta, Daniele Bertini

Journal:

Year:

2003

Language:

english

File:

PDF, 174 KB

english, 2003

24

An Approach to Novel Fused Triazole or Tetrazole Derivatives Starting from Benzimidazo[1,2-a]quinazoline-5(7H)-one and 5,7-Dihydro-5-oxopyrido[3′,2′:5,6]pyrimido[1,2-a]benzimidazole.

Antonio Da Settimo, Giampaolo Primofiore, Federico Da Settimo, Gianluca Pardi, Francesca Simorini, Anna Maria Marini

Journal:

Year:

2003

Language:

english

File:

PDF, 166 KB

english, 2003

25

Synthesis of Novel 1,4-Dihydropyrido[3′,2′:5,6]thiopyrano[4,3-c]pyrazoles and 5H-Pyrido[3′,2′:5,6]thiopyrano[4,3-d]pyrimidines as Potential Antiproliferative Agents.

Giampaolo Primofiore, Anna Maria Marini, Federico Da Settimo, Silvia Salerno, Daniele Bertini, Lisa Dalla Via, Sebastiano Marciani Magno

Journal:

Year:

2004

File:

PDF, 138 KB

2004

26

Synthesis of Pyrimido[1,2-a]benzimidazol-4(10H)-one Derivatives and Evaluation of Their Interactions with DNA.

A. Da Settimo, G. Primofiore, F. Da Settimo, A. M. Marini, S. Taliani, S. Salerno, L. Dalla Via

Journal:

Year:

2004

File:

PDF, 100 KB

2004

27

Synthesis and Benzodiazepine Receptor Affinity of Derivatives of the New Tricyclic Heteroaromatic System Pyrido[3′,2′:5,6]thiopyrano[4,3-c]pyridazin-3(2H,5H)-one.

Giampaolo Primofiore, Federico Da Settimo, Anna Maria Marini, Francesca Simorini, Concettina La Motta, Sabrina Taliani, Sonia Laneri, Letizia Trincavelli, Claudia Martini

Journal:

Year:

2005

File:

PDF, 25 KB

2005

28

ChemInform Abstract: Synthesis and Biological Evaluation of [2′-Oxo-2,3-dihydro-3′H-spiro[chromene-4,5′- [1,3]oxazolidin]-3′yl]acetic Acid Derivatives as Aldose Reductase Inhibitors.

Simona Rapposelli, Frederico Da Settimo, Maria Digiacomo, Concettina La Motta, Annalina Lapucci, Stefania Sartini, Michael Vanni

Journal:

Year:

2011

File:

PDF, 62 KB

2011

29

Highlighting the New Advances in Drug Discovery and Development

Sabrina Taliani, Federico Da Settimo

Journal:

Year:

2008

Language:

english

File:

PDF, 149 KB

english, 2008

30

A Virtual Screening Study of the 18 kDa Translocator Protein using Pharmacophore Models Combined with 3D-QSAR Studies

Tiziano Tuccinardi, Sabrina Taliani, Marusca Bellandi, Federico Da Settimo, Eleonora Da Pozzo, Claudia Martini, Adriano Martinelli

Journal:

Year:

2009

Language:

english

File:

PDF, 404 KB

english, 2009

31

Derivatives of Benzimidazol-2-ylquinoline and Benzimidazol-2-ylisoquinoline as Selective A1 Adenosine Receptor Antagonists with Stimulant Activity on Human Colon Motility

Prof. Barbara Cosimelli, Dr. Sabrina Taliani, Prof. Giovanni Greco, Prof. Ettore Novellino, Dr. Annalisa Sala, Dr. Elda Severi, Prof. Federico Da Settimo, Dr. Concettina La Motta, Dr. Isabella Puglies

Journal:

Year:

2011

Language:

english

File:

PDF, 676 KB

english, 2011

32

A1 adenosine receptor antagonists, 3-aryl[1,2,4]triazino[4,3-a]benzimidazol-4-(10H)-ones (ATBIs) and N-alkyl and N-acyl-(7-substituted-2-phenylimidazo[1,2-a][1,3,5]triazin-4-yl)amines (ITAs): Different recognition of bovine and human binding sites

Federico Da Settimo, Giampaolo Primofiore, Sabrina Taliani, Concettina La Motta, Ettore Novellino, Giovanni Greco, Antonio Lavecchia, Barbara Cosimelli, Manuela Iadanza, Karl-Norbert Klotz, Daniela Tu

Journal:

Drug Development Research

Year:

2004

Language:

english

File:

PDF, 101 KB

english, 2004

33

Synthesis of purinobenzothiazine and pyridothiazinopurine derivatives. Two new heterocyclic ring systems

Antonio Da Settimo, Anna Maria Marini, Giampaolo Primofiore, Federico Da Settimo, Daniele Bertini

Journal:

Journal of Heterocyclic Chemistry

Year:

1998

File:

PDF, 229 KB

1998

34

Synthesis of purinobenzodiazepine and purinobenzotriazocine derivatives, two new heterocyclic ring systems

Antonio Da Settimo, Giampaolo Primofiore, Anna Maria Marini, Federico Da Settimo, Concettina La Motta, Silvia Salerno

Journal:

Journal of Heterocyclic Chemistry

Year:

1999

File:

PDF, 218 KB

1999

35

Synthesis of novel 5H, 11H-pyrido[2′,3′:2,3]thiopyrano[4,3-b]-indoles by fischer-indole cyclization

Antonio Da Settimo, Anna Maria Marini, Giampaolo Primofiore, Federico Da Settimo, Silvia Salerno, Concettina La Motta, Gianluca Pardi, Pier Luigi Ferrarini, Claudio Mori

Journal:

Journal of Heterocyclic Chemistry

Year:

2000

File:

PDF, 222 KB

2000

36

Synthesis of a novel purine-containing heterocyclic ring system: 8,10-Dimethylindolo[2′,3′:5,6][1,2,4]triazino[4,3-f]purine-9,11(8H, 10H, 13H)-dione

Antonio Da Settimo, Giampaolo Primofiore, Federico Da Settimo, Francesca Simorini, Anna Maria Marini, Concettina La Motta, Sabrina Taliani

Journal:

Journal of Heterocyclic Chemistry

Year:

2000

File:

PDF, 282 KB

2000

37

Facile synthesis of 3-substituted [1,2,4]triazino[3,4-f]purine-4,6,8-trione derivatives

Federico Da Settimo, Anna Maria Marini, Gianluca Pardi, Giampaolo Primofiore, Silvia Salerno, Francesca Simorini

Journal:

Journal of Heterocyclic Chemistry

Year:

2001

Language:

english

File:

PDF, 56 KB

english, 2001

38

Synthesis of novel pyrido[3′,2′:5,6]thiopyrano[3,2-b]indol-5(6H)-ones and 6H-pyrido[3′,2′:5,6]thiopyrano[4,3-b]quinolines, two new heterocyclic ring systems

Antonio Da Settimo, Anna María Marini, Giampaolo Primofiore, Federico Da Settimo, Silvia Salerno, Francesca Simorini, Gianluca Pardi, Concettina La Motta, Daniele Bertini

Journal:

Journal of Heterocyclic Chemistry

Year:

2002

Language:

english

File:

PDF, 53 KB

english, 2002

39

An approach to novel fused triazole or tetrazole derivatives starting from benzimidazo[1,2-a]quinazoline-5(7H)-one and 5,7-dihydro-5-oxopyrido[3′,2′:5,6]pyrimido[1,2-a]benzimidazole

Antonio Da Settimo, Giampaolo Primofiore, Federico Da Settimo, Gianluca Pardi, Francesca Simorini, Anna Maria Marini

Journal:

Journal of Heterocyclic Chemistry

Year:

2002

Language:

english

File:

PDF, 64 KB

english, 2002

40

Synthesis of novel 1,4-dihydropyrido[3′,2′:5,6]thiopyrano[4,3-c]-pyrazoles and 5H-pyrido[3′,2′:5,6]thiopyrano[4,3-d]pyrimidines as potential antiproliferative agents

Giampaolo Primofiore, Anna Maria Marini, Federico Da Settimo, Silvia Salerno, Daniele Bertini, Lisa Dalla Via, Sebastiano Marciani Magno

Journal:

Journal of Heterocyclic Chemistry

Year:

2003

Language:

english

File:

PDF, 98 KB

english, 2003

41

Synthesis of pyrimido[1,2-a]benzimidazol-4(10H)-one derivatives and evaluation of their interactions with DNA

A. Da Settimo, G. Primofiore, F. Da Settimo, A. M. Marini, S. Taliani, S. Salerno, L. Dalla Via

Journal:

Journal of Heterocyclic Chemistry

Year:

2003

Language:

english

File:

PDF, 64 KB

english, 2003

42

Synthesis and antiproliferative evaluation of new aryl substituted pyrido[3′,2′:5,6]thiopyrano[4,3-c]pyrazoles

G. Primofiore, A. M. Marini, S. Salerno, F. Da Settimo, D. Bertini, L. Dalla Via

Journal:

Journal of Heterocyclic Chemistry

Year:

2005

Language:

english

File:

PDF, 97 KB

english, 2005

43

Synthesis of New Heterocyclic Ring Systems via [1,3,5]Triazino[1,2-a]benzimidazole Derivatives

Giampaolo Primofiore, Federico Da Settimo, Gianluca Pardi, Francesca Simorini, Concettina La Motta, Silvia Salemo, Sabrina Taliani, Anna Maria Marini

Journal:

Journal of Heterocyclic Chemistry

Year:

2005

Language:

english

File:

PDF, 124 KB

english, 2005

44

Synthesis and in vitro antiproliferative activity of new substituted benzo[3′,2′:5,6]thiopyrano[4,3-d]pyrimidines

Anna Maria Marini, Federico Da Settimo, Silvia Salerno, Concettina La Motta, Francesca Simorini, Sabrina Taliani, Daniele Bertini, Ornella Gia, Lisa Dalla Via

Journal:

Journal of Heterocyclic Chemistry

Year:

2008

Language:

english

File:

PDF, 261 KB

english, 2008

45

The nitration of some phenyl substituted indoles

A. Da Settimo, M.F. Saettone

Journal:

Year:

1965

Language:

english

File:

PDF, 655 KB

english, 1965

46

N-(Indol-3-ylglyoxylyl)methionine derivatives: preparation and gastric anti-secretory activity

Antonio Da Settimo, Giampaolo Primofiore, Anna Maria Marini, Pier Luigi Ferrarini, JosèSebastian Franzone, Rocco Cirillo, Maria Camilla Reboani

Journal:

European Journal of Medicinal Chemistry

Year:

1988

Language:

english

File:

PDF, 408 KB

english, 1988

47

N-(Indol-3-ylglyoxylyl)dopamine derivatives: preparation and anti-depressant activity

Giampaolo Primofiore, Anna Maria Marini, Federico da Settimo, JosèSebastian Franzone, Ugo Mason, Maria Camilla Reboani, Rocco Cirillo

Journal:

European Journal of Medicinal Chemistry

Year:

1988

Language:

english

File:

PDF, 364 KB

english, 1988

48

Reinvestigation of reductive butylation of aminophthalimides: new compounds with local anesthetic activity

Antonio da Settimo, Giampaolo Primofiore, Pier L Ferrarini, Maria Ferretti, Pier L Barili, Natale Tellini, Pietro Bianchini

Journal:

European Journal of Medicinal Chemistry

Year:

1989

Language:

english

File:

PDF, 742 KB

english, 1989

49

Synthesis and β-blocking activity of (E)- and (Z)-iminoethers of 1,8-naphthyridine. Potential antihypertensive agents. 4

PL Ferrarini, C Mori, G Primofiore, A Da Settimo, MC Breschi, E Martinotti, P Nieri, MA Ciucci

Journal:

European Journal of Medicinal Chemistry

Year:

1990

Language:

english

File:

PDF, 582 KB

english, 1990

50

1-substituted 2-benzylaminobenzimidazole derivatives: compounds with H1-antihistaminic activity

A Da Settimo, G Primofiore, F Da Settimo, L Calzolari, P Cazzulani, A Passoni, O Tofanetti

Journal:

European Journal of Medicinal Chemistry

Year:

1992

Language:

english

File:

PDF, 539 KB

english, 1992